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Black Market Testosterone
by RaverDyke, Trans-Health.com

(The Gender Centre advise that this article may not be current and as such certain content, including
but not limited to persons, contact details and dates may not apply. Where legal authority or medical related matters are
cited, responsibility lies with the reader to obtain the most current relevant legal authority and/or medical
publication.)
Counterfeit androgens are a huge and profitable business for many unscrupulous people.
Do not buy testosterone from the black market, especially from body builders. They will probably
rip you off, and there's absolutely no telling what you will get, if it will contain what it says, or even if it is sanitary or sterile.
Counterfeit androgens are a huge and profitable business for many unscrupulous people. What they give you might be dangerous, I'm not
kidding.
Below I describe four androgens and a few other drugs that might be of interest to
F.T.M. guys. Remember that 250mg of one testosterone ester is not the same as 250mg of
another testosterone ester, nor is it the same as 250mg of another androgen. I won't make specific dosage recommendations: that's up to
your physician.
Testosterone
Testosterone is the F.T.M.s androgen of choice for a variety of reasons. It has
excellent androgenic and anabolic properties, and is the substance that is produced naturally within your body. It does have a 5αR
metabolite and an aromatase metabolite, so one should consider adding an anti-estrogenic agent if one is supplementing with
supraphysiological doses of the drug. If you are prone to hair loss and/or male pattern baldness, you should also consider a 5αR
inhibitor. Physicians specializing in hair loss can usually help you find an appropriate one. There are several different testosterone
drugs, including testosterone cypionate (Depo-testosterone), testosterone enanthate (Testoviron/Delatestryl), testosterone propionate and
testosterone decanoate. Testosterone cypionate and testosterone enanthate are the most common testosterone esters used by
F.T.M.s. One possibility that F.T.M.s
should consider is a drug called Sustanon 250, which is an injectable drug containing 250mg of four different testosterone esters. It might
not be available in your country. Organon is reputable manufacturer of Sustanon 250, but there's a whole bunch of fake Sustanon out there.
Buy it from a reputable pharmacy. Omnadren 250 is a drug similar to Sustanon 250, but with one different ester that reduces the overall
half life by a few days. Omnadren is also faked quite frequently.
Nandrolone
At first glance nandrolone might seem to be a weird substance. It resembles both an androgen and an estrogen, but it has reasonably high
anabolic effects. It is known to be a progestin, which might cause some undesirable effects in an
F.T.M. guy. Nevertheless, it is a reasonable choice, especially for guys who are concerned
about hair loss or specifically about gaining muscle size. By far the most common nandrolone drug is the injectable Deca Durabolin, or
nandrolone decanoate. This is without a doubt the most commonly counterfeited androgen, so definitely don't buy it off of the street.
Trenbolone
I think this androgen rocks. It seems to cause the fewest negative side effects and the maximum positive effects. Pound for pound it
seems to be almost three times as effective as testosterone. It has no metabolic pathway to estrogens, and seems to have reasonably little
negative effect on hair loss. Unfortunately it is very hard to get in most countries. One possibility is the drug Parabolan (trenbolone
cyclohexylmethylcarbonate), an oil-based injectable. There are some agricultural drugs containing trenbolone, but ... well, they're not
made for human use. Same drug, possibly fewer quality controls during the manufacturing process. And if you buy this on the black market
(assuming that what you buy even contains trenbolone, and that's quite an assumption to make) you're probably buying something that someone
whipped up in his basement after extracting trenbolone acetate from cattle implants. Most of these people know and care very little about
making the drug safe. But Good Gravy, if you can find trenbolone then you should definitely ask your doctor for a prescription.
Methenolone
This is a weaker androgen, but a reasonable choice for F.T.M. guys because it does not
metabolize to an estrogen. It might increase the rate of hair loss, but seems to be less aggressive in this regard than testosterone.
Primobolan Depot (methenolone enanthate) is the most common injectable preparation of methenolone. Primobolan is expensive.
Other Androgens
There are quite a few oral androgens that I'm just not going to mention. Suffice to say that you should stay away from them if you can
find injectables. If you are seeing a physician, just have him prescribe an injectable and show you how to inject it (or have him inject it
for you).
Clomiphene
Clomiphene seems to be a very effective anti-estrogenic compound. It is not an androgen. It is most commonly used in the treatment of
breast cancer. It is an oral drug, but as it is not an oral androgen it does not have hepatotoxic effects. The most common drug preparation
of clomiphene is called Clomid (clomiphene citrate). It is widely available around the world.
Aminoglutethimide
This is a drug that inhibits the action of aromatase, the enzyme that converts androgens to estrogens. At higher dosages, through
another mechanism, it can inhibit the production of cortisol. This might sound good (cortisol is catabolic) but you need normal cortisol
levels to be healthy. If you're going to take aminoglutethimide, don't take a lot of it, and have your cortisol levels checked regularly.
The brand name for it is Cytadren. There are better anti-estrogenic choices such as tamoxifen and clomiphene, so really, don't bother with
it.
Anastrozole
This compound works like aminoglutethimide in that it blocks the aromatization of androgens to estrogens, but it does not seem to have
the same effects on cortisol. Its brand name is Arimidex. It is expensive but effective. I still think tamoxifen and clomiphene are better
choices for anti-estrogens.
Tamoxifen
Tamoxifen is quite similar to clomphene. Most readily available under the brand name Nolvadex, and like clomiphene it blocks estrogen
receptors in some tissues and activates them in others. (However, this activation in reality blocks the estrogenic effects anyway, so no
worries.)
To summarize, keep all of this in mind the next time you talk to your physician:
- They can probably double, triple or even quadruple your dosage of testosterone with great results and few negative effects,
especially for periods of a few weeks or months.
- There are drugs available that reduce estrogenic effects. You should consider them, especially if you are using
testosterone.
- There are other androgens available besides testosterone.
- You should have your lipid, testosterone, estrogen and liver levels, as well as your blood pressure, checked regularly.
Glossary
- Anabolic: An effect that increases growth. For F.T.M.
purposes this usually refers to muscle growth, and should more specifically be described as "muscle anabolism."
- Androgenic: A "masculinizing" effect such as increased body hair growth.
- 17-alpha alkylated: A steroid that has an alkyl group attached at the 17alpha position.
- Acute: A state or condition that comes on rapidly and disappears within a short amount of time.
- Ester: In chemistry, an organic compound in which an oxygen is bonded to carbon atom(s). In practical terms
relevant to our discussion of androgens, esters of drugs are more soluble in oil (important for many injectable drugs) and
longer-acting because it appears that the body must remove the ester chain before the compound can act at androgen receptors.
- Half-life: - For our purposes, the amount of time it takes for a substance to be metabolically reduced to one
half of its original concentration.
- Metabolic: An action that takes place inside the body.
- Oral: A delivery mechanism that involves taking a drug by mouth.
- Supraphysiological: Dosages that are greater than what the "normal, healthy" body will produce
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